Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM82423'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Mainz
Curated by ChEMBL
University of Mainz
Curated by ChEMBL
Affinity DataKi: 0.269nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Mainz
Curated by ChEMBL
University of Mainz
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Inhibition of [3H]NMS binding to rat heart Muscarinic acetylcholine receptor M2Checked by AuthorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Mainz
Curated by ChEMBL
University of Mainz
Curated by ChEMBL
Affinity DataKi: 0.302nMAssay Description:Displacement of [3H]N-methylscopolamine chloride from human cloned muscarinic M2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair