Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M3' and Ligand = 'BDBM50581208'
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))TBA
LigandPNGBDBM50581208(CHEMBL5076535)copy SMILES
Affinity DataKi:  12.6nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN48WCPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))TBA
LigandPNGBDBM50581208(CHEMBL5076535)copy SMILES
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-N-methyl Scopolamine Chloride from human M3 receptor membranes incubated for 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN48WCPubMed
LigandPNGBDBM50581208(CHEMBL5076535)copy SMILES
Affinity DataIC50: 79nMAssay Description:Antagonist activity at muscarinic M3 receptor in rat trachea assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN48WCPubMed
LigandPNGBDBM50581208(CHEMBL5076535)copy SMILES
Affinity DataIC50: 79.4nMAssay Description:Antagonist activity at muscarinic M3 receptor in rat trachea assessed as inhibition of carbachol-induced contractionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN48WCPubMed