Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50323693'
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50323693(3-amino-N-benzyl-4,6-dimethylthieno[2,3-b]pyridine...)copy SMILEScopy InChI
Affinity DataEC50:  1.30E+3nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 15 nM acetylcholine-induced calciu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50N55PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50323693(3-amino-N-benzyl-4,6-dimethylthieno[2,3-b]pyridine...)copy SMILEScopy InChI
Affinity DataEC50:  0.000693nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2251GKRPCBioAssay