Found 5 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50403547'
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataKi: 0.520nMAssay Description:Displacement of [3H]NMS from rat recombinant muscarinic M4 receptor expressed in CHO cells after 2 hrs by microplate scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataKi: 0.520nMAssay Description:Displacement of [3H]NMS from rat recombinant muscarinic M4 receptor expressed in CHO cells after 2 hrs by microplate scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Displacement of [3H]NMS from rat muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataKi: 1.39nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M4 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Walter Reed Army Institute of Research
Curated by ChEMBL
Walter Reed Army Institute of Research
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-4-DAMP from human muscarinic M4 receptor expressed in BHK-21 cellsMore data for this Ligand-Target Pair