Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50403547'
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)copy SMILEScopy InChI
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]NMS from rat recombinant muscarinic M4 receptor expressed in CHO cells after 2 hrs by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50N55PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)copy SMILEScopy InChI
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]NMS from rat recombinant muscarinic M4 receptor expressed in CHO cells after 2 hrs by microplate scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50N55PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
DVanderbilt Program in Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)copy SMILEScopy InChI
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]NMS from rat muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ095ZPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Walter Reed Army Institute of Research

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)copy SMILEScopy InChI
Affinity DataKi:  1.39nMAssay Description:Displacement of [3H] N-methylscopolamine from human muscarinic M4 receptor expressed in CHOK1 cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92F6XPubMedDrugBank
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Walter Reed Army Institute of Research

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-4-DAMP from human muscarinic M4 receptor expressed in BHK-21 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765G9KPubMedDrugBank