Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM50423967'
TargetMuscarinic acetylcholine receptor M4(RAT)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423967(CHEMBL2057417)copy SMILEScopy InChI
Affinity DataEC50:  176nMAssay Description:Positive allosteric modulation of rat muscarinic M4 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29Z8SPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423967(CHEMBL2057417)copy SMILEScopy InChI
Affinity DataEC50:  56nMAssay Description:Positive allosteric modulation of human muscarinic M4 receptor expressed in CHO-K1 cells assessed as leftward shift in acetylcholine response treated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29Z8SPubMed