Found 5 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Ligand = 'BDBM50403547'
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of South Florida
Curated by ChEMBL
University of South Florida
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]QNB from muscarinic acetylcholine M5 receptor after 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataKi: 0.860nMAssay Description:Displacement of [3H]NMS from rat recombinant muscarinic M5 receptor expressed in CHO cells after 2 hrs by microplate scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of South Florida
Curated by ChEMBL
University of South Florida
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-4-DAMP from human muscarinic M5 receptor expressed in BHK-21 cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of South Florida
Curated by ChEMBL
University of South Florida
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]NMS from human muscarinic acetylcholine receptor subtype 5 expressed in CHO cell membranes by scintillation counting methodMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M5(RAT)
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
DVanderbilt Program in Drug Discovery
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]NMS from rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair