Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Neuroepithelial cell-transforming 1' and Ligand = 'BDBM50337910'
TargetNeuroepithelial cell-transforming 1(Rat)
SUNOVION PHARAMCEUTICALS INC.

US Patent
LigandPNGBDBM50337910((+/-)-1-(1-(3,4-dichlorophenyl)cyclohexyl)-N-methy...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Quantification of norepinephrine uptake was performed using synaptosomes isolated in a 0.32 M sucrose buffer from a male Wistar rat hypothalamus. The...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP77BXUS Patent
TargetNeuroepithelial cell-transforming 1(Rat)
SUNOVION PHARAMCEUTICALS INC.

US Patent
LigandPNGBDBM50337910((+/-)-1-(1-(3,4-dichlorophenyl)cyclohexyl)-N-methy...)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Quantification of norepinephrine uptake was performed using synaptosomes isolated in a 0.32 M sucrose buffer from a male Wistar rat hypothalamus. The...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP77BXUS Patent
TargetNeuroepithelial cell-transforming 1(Rat)
SUNOVION PHARAMCEUTICALS INC.

US Patent
LigandPNGBDBM50337910((+/-)-1-(1-(3,4-dichlorophenyl)cyclohexyl)-N-methy...)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Quantification of norepinephrine uptake was performed using synaptosomes isolated in a 0.32 M sucrose buffer from a male Wistar rat hypothalamus. The...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP77BXUS Patent
TargetNeuroepithelial cell-transforming 1(Rat)
SUNOVION PHARAMCEUTICALS INC.

US Patent
LigandPNGBDBM50337910((+/-)-1-(1-(3,4-dichlorophenyl)cyclohexyl)-N-methy...)copy SMILEScopy InChI
Affinity DataIC50: 74nMAssay Description:Quantification of norepinephrine uptake was performed using synaptosomes isolated in a 0.32 M sucrose buffer from a male Wistar rat hypothalamus. The...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XP77BXUS Patent