Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Neuromedin-B receptor' and Ligand = 'BDBM50295231'
TargetNeuromedin-B receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50295231((+)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24WG8PubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50295231((+)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24WG8PubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50295231((+)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)copy SMILEScopy InChI
Affinity DataIC50: 580nMAssay Description:Antagonist activity at human neuromedin B receptor transfected in HEK293 cells assessed as inhibition of 1 nM neuromedin B-induced myo-[3H]inositol p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24WG8PubMed
TargetNeuromedin-B receptor(Homo sapiens (Human))
Amgen Inc.

Curated by ChEMBL
LigandPNGBDBM50295231((+)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24WG8PubMed