Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Neuromedin-K receptor' and Ligand = 'BDBM50284763'
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284763(1-(3-Benzyl-pyrrolidin-1-yl)-2-(1H-indol-3-yl)-eth...)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [3H]senktide to Tachykinin receptor 3 in the guinea pig cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD1ZDC
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50284763(1-(3-Benzyl-pyrrolidin-1-yl)-2-(1H-indol-3-yl)-eth...)copy SMILEScopy InChI
Affinity DataIC50: 4.40E+3nMAssay Description:Binding affinity towards Tachykinin receptor 3 using [125I]-[Mephe7] NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4C27