Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Neuromedin-K receptor' and Ligand = 'BDBM50341110'
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341110((4-(2-methoxyphenyl)piperazin-1-yl)(3-(pyridin-2-y...)copy SMILEScopy InChI
Affinity DataKi:  3.60E+3nMAssay Description:Displacement [3H]SB-222200 from of human recombinant NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
Euroscreen SA

Curated by ChEMBL
LigandPNGBDBM50341110((4-(2-methoxyphenyl)piperazin-1-yl)(3-(pyridin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at human recombinant NK3 receptor expressed in CHO cells assessed as inhibition of NKB-induced increase of intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56K16PubMed