Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Neuromedin-U receptor 2' and Ligand = 'BDBM50291674'
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50291674(CHEMBL4159176)copy SMILEScopy InChI
Affinity DataIC50: 429nMAssay Description:Displacement of [3H]-NMU-8 from human NMUR2 expressed in HEK293 cell membranes after 3 hrs by microscintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50291674(CHEMBL4159176)copy SMILEScopy InChI
Affinity DataEC50:  382nMAssay Description:Agonist activity at human NMUR2 expressed in HEK293 cells assessed as induction of IP3 levels using myo-[2-3H(N)]-inositol after 60 mins by SPA-based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91JPPubMed