Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/beta-2' and Ligand = 'BDBM50246823' TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies
Curated by ChEMBL
Torrey Pines Institute for Molecular Studies
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Torrey Pines Institute for Molecular Studies
Curated by ChEMBL
Torrey Pines Institute for Molecular Studies
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat alpha4beta2 nAChR expressed in HEK cells assessed as inhibition of epibatidine-induced membrane potential preincubated for...More data for this Ligand-Target Pair
