Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/beta-2' and Ligand = 'BDBM50257941'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50257941(7-(pyridin-3-yl)-1,7-diazaspiro[4.4]nonane | CHEMB...)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50257941(7-(pyridin-3-yl)-1,7-diazaspiro[4.4]nonane | CHEMB...)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-epibatidine from human nAChR alpha4beta2 expressed in human SH-EP1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X58W1PubMed