Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4' and Ligand = 'BDBM50472282'
TargetNeuronal acetylcholine receptor subunit alpha-4(Gallus gallus)
Gifu University
Curated by ChEMBL
Gifu University
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Mus musculus)
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of [3H]nicotine binding to alpha4 nicotinic acetylcholine receptor in Mus musculus (mouse) M10 cells co-expressing beta2 nicotinic acetylc...More data for this Ligand-Target Pair