Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Neuropeptide FF receptor 1' and Ligand = 'BDBM50060728'
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
CNRS/IPBS (Institut de Pharmacologie et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50060728((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Binding affinity to human NPFF1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3BVGPubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
CNRS/IPBS (Institut de Pharmacologie et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50060728((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]NPVF from human NPFF1 expressed in CHO cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3BVGPubMed
TargetNeuropeptide FF receptor 1(Homo sapiens (Human))
CNRS/IPBS (Institut de Pharmacologie et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50060728((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...)copy SMILEScopy InChI
Affinity DataKd:  20.9nMAssay Description:Competitive antagonist activity at human NPFF1 receptor expressed in COS1 cells assessed as inhibition of NPVF-induced [3H]inositol phosphate accumul...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974PVPubMed