Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Neuropeptide Y receptor type 1' and Ligand = 'BDBM50500157'
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
CNRS/IPBS (Institut de Pharmacologie et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500157(CHEMBL4299523)copy SMILEScopy InChI
Affinity DataKi:  0.410nMAssay Description:Displacement of (R)-Na-Diphenylacetyl-Nomega[2-([2,3-3H]-propionylamino)ethyl]aminocarbonyl (4-hydroxybenzyl)-argininamide from NPY1R in human SK-N-M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3BVGPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
CNRS/IPBS (Institut de Pharmacologie et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500157(CHEMBL4299523)copy SMILEScopy InChI
Affinity DataKi:  0.420nMAssay Description:Displacement of (R)-Na-Diphenylacetyl-Nomega[2-([2,3-3H]-propionylamino)ethyl]aminocarbonyl (4-hydroxybenzyl)-argininamide from NPY1R in human SK-N-M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3BVGPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
CNRS/IPBS (Institut de Pharmacologie et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500157(CHEMBL4299523)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]propionyl-pNPY from NPY1R in HEL cells after 60 to 90 mins by flow cytometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3BVGPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
CNRS/IPBS (Institut de Pharmacologie et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500157(CHEMBL4299523)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]UR-MK136 from NPY1R in human SK-N-MC cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3BVGPubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
CNRS/IPBS (Institut de Pharmacologie et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500157(CHEMBL4299523)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Displacement of (R)-Na-Diphenylacetyl-Nomega[2-([2,3-3H]-propionylamino)ethyl]aminocarbonyl (4-hydroxybenzyl)-argininamide from NPY1R in human SK-N-M...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN3BVGPubMed