Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Nicotinamide phosphoribosyltransferase' and Ligand = 'BDBM50236219'
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50236219(CHEMBL4066091)copy SMILEScopy InChI
Affinity DataIC50: 7.80nMAssay Description:Inhibition of NAMPT in human Jurkat T cells assessed as reduction in NAD levelsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ63TKPubMed
TargetNicotinamide phosphoribosyltransferase(Mus musculus)
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50236219(CHEMBL4066091)copy SMILEScopy InChI
Affinity DataIC50: 8.10nMAssay Description:Inhibition of recombinant mouse NAMPT expressed in bacterial expression system using nicotinamide as substrate after 1 hr by fluorescence based NMNAT...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ63TKPubMed