Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Nischarin' and Ligand = 'BDBM50179395'
TargetNischarin(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding affinity for imidazoline receptor I-2 in rabbit kidney homogenate (relative to [3H]-Idazoxan radioligand)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB48G9PubMed
TargetNischarin(RAT)TBA
LigandPNGBDBM50179395(CHEMBL14640)copy SMILEScopy InChI
Affinity DataKi:  692nMAssay Description:Binding affinity to I1 imidazoline binding site in Rattus norvegicus (rat) PC12 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2KNG
TargetNischarin(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)copy SMILEScopy InChI
Affinity DataKi:  708nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6NSWPubMed
TargetNischarin(RAT)TBA
LigandPNGBDBM50179395(CHEMBL14640)copy SMILEScopy InChI
Affinity DataKi:  708nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ89J3PubMed