Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-gamma' and Ligand = 'BDBM50035915'
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50035915(CHEMBL3361058)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]25-hydroxycholesterol from human RORc-LBD expressed in bacterial expression system after 3 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V8FPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50035915(CHEMBL3361058)copy SMILEScopy InChI
Affinity DataEC50:  22nMAssay Description:Inverse agonist activity at N-terminal 6xHis-tagged human RORc ligand binding domain expressed in bacterial expression system assessed as inhibition ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V8FPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery Ltd.

Curated by ChEMBL
LigandPNGBDBM50035915(CHEMBL3361058)copy SMILEScopy InChI
Affinity DataEC50:  19nMAssay Description:Inverse agonist activity at GAL4-fused human RORc expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125V8FPubMed