Affinity DataEC50: <500nMAssay Description:Agonist activity at His tagged RORgammat LBD (unknown origin) expressed in baculovirus infected sf9 cells assessed as biotinylated-LXXLL peptide coac...More data for this Ligand-Target Pair
Affinity DataEC50: 324nMAssay Description:Agonist activity at human ROR-gamma LBD expressed in HEK293 cells assessed as transcriptional activity in presence of ursolic acid by Gal4-luciferase...More data for this Ligand-Target Pair
Affinity DataEC50: 223nMAssay Description:Agonist activity at human His-tagged RORgamma-LBD expressed in Sf9 cells assessed as inhibition of N-terminal biotinylated co-activator SRC1 recruitm...More data for this Ligand-Target Pair
Affinity DataEC50: <500nMAssay Description:In vivo inhibition of leutenising hormone in rats.More data for this Ligand-Target Pair