Found 1 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 2' and Ligand = 'BDBM50054245'
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
City of Hope National Medical Center
Curated by ChEMBL
City of Hope National Medical Center
Curated by ChEMBL
Affinity DataEC50: 4.95E+3nMAssay Description:Agonist activity at PXR (unknown origin) expressed in human HepG2 cells assessed as induction of CYP3A4 transactivation after 16 hrs by luciferase re...More data for this Ligand-Target Pair