BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with Target = 'POU domain, class 2, transcription factor 2' and Ligand = 'BDBM50228403'

POU domain, class 2, transcription factor 2(Homo sapiens (Human))
Nippon Boehringer Ingelheim Co., Ltd.

Curated by ChEMBL

BDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)copy SMILEScopy InChI

IC50: 8.00E+4nMAssay Description:Inhibition of OCT2 (unknown origin) expressed in HEK293 cells assessed as reduction of [14C]metformin substrate uptake at 100 uM by liquid scintillat...More data for this Ligand-Target Pair

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Details Article
BindingDB Entry DOI: 10.7270/Q2QC0574PubMed