Found 1 Enz. Inhib. hit(s) with Target = 'Peptidyl-prolyl cis-trans isomerase FKBP1A/Ryanodine receptor 1' and Ligand = 'BDBM50191286'
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A/Ryanodine receptor 1(Homo sapiens (Human))
University of California
Curated by ChEMBL
University of California
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Agonist like activity at skeletal junction sarcoplasmic reticulum RyR1/FKBP12 complex assessed as increase in [3H]ryanodine bindingMore data for this Ligand-Target Pair