Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Peptidyl-prolyl cis-trans isomerase FKBP1A/Ryanodine receptor 1' and Ligand = 'BDBM50191286'
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A/Ryanodine receptor 1(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50191286(Bastadin-5 | CHEMBL439151 | bastadin 5)copy SMILEScopy InChI
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist like activity at skeletal junction sarcoplasmic reticulum RyR1/FKBP12 complex assessed as increase in [3H]ryanodine bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0WNDPubMed