Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50172806'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
CNRS UMR 6052
Curated by ChEMBL
CNRS UMR 6052
Curated by ChEMBL
Affinity DataKi: 718nMAssay Description:Binding affinity for human PPAR gamma construct expressed in bacteria with 3[H] rosiglitazoneMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
CNRS UMR 6052
Curated by ChEMBL
CNRS UMR 6052
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro effective concentration against human peroxisome proliferator activated receptor gamma/Gal4 in cell-based transactivation assayMore data for this Ligand-Target Pair