Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform' and Ligand = 'BDBM50436459'
LigandPNGBDBM50436459(CHEMBL2396661)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibition of N-terminal His6-tagged human recombinant full length PI3Kdelta co-expressed with human recombinant full length P85alpha in baculovirus ...More data for this Ligand-Target Pair
LigandPNGBDBM50436459(CHEMBL2396661)copy SMILEScopy InChI
Affinity DataIC50: 383nMAssay Description:Inhibition of human PI3K p110delta/p85alpha using PIP2 as substrate in presence of ATP measured after 40 mins by HTRF assayMore data for this Ligand-Target Pair