Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform' and Ligand = 'BDBM50193023'
LigandPNGBDBM50193023(CHEMBL3898901 | US11155556, No. 5)copy SMILEScopy InChI
Affinity DataIC50: 728nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193023(CHEMBL3898901 | US11155556, No. 5)copy SMILEScopy InChI
Affinity DataIC50: 730nMAssay Description:Inhibition of human PI3Kalpha (R108 to N1068 residues) expressed in mammalian expression system incubated for 60 mins by ADAPTA assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P91B0PubMed