Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform' and Ligand = 'BDBM50394841'
LigandPNGBDBM50394841(CHEMBL2165004 | US8772480, 228)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Inhibition of human N-terminal poly-His tagged-PI3Kalpha expressed in Sf9 baculovirus system co-expressing p85alpha after 20 mins by AlphaScreen assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4QSJPubMed
LigandPNGBDBM50394841(CHEMBL2165004 | US8772480, 228)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:The PI3K AlphaScreen assay (PerkinElmer, Waltham, Mass.) measures the activity of a panel of four phosphoinositide 3-kinases: PI3Kalpha, PI3Kbeta, PI...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V123FJUS Patent