Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform' and Ligand = 'BDBM50534995'
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50534995(CHEMBL4095008)copy SMILEScopy InChI
Affinity DataIC50: 396nMAssay Description:Inhibition of PI3Kbeta (unknown origin) expressed in baculovirus expression system by kinase-glo luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9F98PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50534995(CHEMBL4095008)copy SMILEScopy InChI
Affinity DataIC50: 565nMAssay Description:Inhibition of full length His-tagged human recombinant PI3Kbeta expressed in baculovirus by select screen kinase profiling assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9F98PubMed