Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform' and Ligand = 'BDBM413450'
LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of AlexaFluor-labeled tracer 236 binding to recombinant full-length human His-tagged p110gamma expressed in baculovirus expression system ...More data for this Ligand-Target Pair
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LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 363nMMore data for this Ligand-Target Pair
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LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of PI3Kgamma in mouse RAW264 cells assessed as reduction in C5a anaphylatoxin trifluoroacetate salt-induced AKT phosphorylation at T208 re...More data for this Ligand-Target Pair
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