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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM27559'
Target
Poly [ADP-ribose] polymerase 1
(Homo sapiens (Human))
KuDOS Pharmaceuticals Ltd.
Ligand
BDBM27559
(4-({4-fluoro-3-[(4-methylpiperazin-1-yl)carbonyl]p...)
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Affinity Data
IC50: 13nM
pH: 7.4 T: 2°C
Assay Description:
A FlashPlate scintillation proximity assay has been developed to identify inhibitors of PARP-1. The mechanism of action of the assay requires the bin...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
antibodypedia
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Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BP014T
PubMed