Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50335640'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Cylene Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335640(4-Oxo-4,5-dihydrothieno[3,2-c]quinoline-7-carboxyl...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of PARP1 by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67H7NPubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Cylene Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335640(4-Oxo-4,5-dihydrothieno[3,2-c]quinoline-7-carboxyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21N857Q