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Compile Data Set for Download or QSAR
Found
1
Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase tankyrase-1' and Ligand = 'BDBM50522353'
Target
Poly [ADP-ribose] polymerase tankyrase-1
(Homo sapiens (Human))
RIKEN
Curated by
ChEMBL
Ligand
BDBM50522353
(CHEMBL4441713)
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Affinity Data
IC50: 6.40nM
Assay Description:
Inhibition of recombinant human N-terminal TEV cleavage site-fused/FLAG-poly his-tagged TNKS SAM-PARP domain (1024 to 1327 residues) expressed in Esc...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2S46WC3
PubMed
PDB
3D Structure (crystal)