Found 1 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase tankyrase-2' and Ligand = 'BDBM50439825' TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Bath
Curated by ChEMBL
University of Bath
Curated by ChEMBL
Affinity DataIC50: 133nMAssay Description:Inhibition of N-terminal GST-tagged human TNKS-2 (849 to 1166 residues) expressed in in insect sf21 cells preincubated for 2 hrs followed by substrat...More data for this Ligand-Target Pair
3D Structure (crystal)