Found 2 Enz. Inhib. hit(s) with Target = 'Polyunsaturated fatty acid 5-lipoxygenase' and Ligand = 'BDBM50530377'
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Universit£ de Moncton
Curated by ChEMBL
Universit£ de Moncton
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of 5-LO in human PMNL cells assessed as reduction in leukotriene formation preincubated for 5 mins followed by thapsigargin stimulation me...More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
Universit£ de Moncton
Curated by ChEMBL
Universit£ de Moncton
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of 5-LO in human PMNL cells assessed as reduction in leukotriene formation preincubated for 5 mins followed by thapsigargin stimulation me...More data for this Ligand-Target Pair