Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 3' and Ligand = 'BDBM50158216'
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50158216(Aceticacid(R)-1-{(4R,4aR,5S,6R,6aR,11bS)-4,5,6-tri...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of voltage-gated potassium channel subunit Kv1.3 in chinese hamster ovary cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0281PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50158216(Aceticacid(R)-1-{(4R,4aR,5S,6R,6aR,11bS)-4,5,6-tri...)copy SMILEScopy InChI
Affinity DataIC50: 29.2nMAssay Description:Inhibitory activity against voltage-gated potassium channel subunit Kv1.3 of human T cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP0281PubMed