Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 3' and Ligand = 'BDBM50279106'
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4X5NPubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Kv1.3 expressed in mouse L929 cells exposed to depolarizing step pulses from -80 mV to +40 mV by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4JXWPubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4B38PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of human Kv1.3 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2668GT4PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)copy SMILEScopy InChI
Affinity DataIC50: 740nMAssay Description:Inhibition of human Kv1.3 ion channel expressed in CGE22 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7VW2PubMed