Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily H member 2' and Ligand = 'BDBM50344942'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Kosan Biosciences, Inc.

Curated by ChEMBL
LigandPNGBDBM50344942(CHEMBL532 | E-MYCIN E | ERYTHROMYCIN | ERYTHROMYCI...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of human ERG expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C1XT1PubMedDrugBank
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Kosan Biosciences, Inc.

Curated by ChEMBL
LigandPNGBDBM50344942(CHEMBL532 | E-MYCIN E | ERYTHROMYCIN | ERYTHROMYCI...)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibitory concentration against IKr potassium channelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q208661KPubMedDrugBank