Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily KQT member 2' and Ligand = 'BDBM50131898'
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50131898((E)-N-[1-((S)-4-Fluoro-3-morpholin-4-yl-phenyl)-et...)copy SMILEScopy InChI
Affinity DataEC50:  1.55E+3nMAssay Description:Effective concentration against Potassium voltage gated channel, KQT-like subfamily, member 2 expressed in SH-SY5Y human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RJ4K66PubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50131898((E)-N-[1-((S)-4-Fluoro-3-morpholin-4-yl-phenyl)-et...)copy SMILEScopy InChI
Affinity DataEC50:  1.20E+3nMAssay Description:Effective concentration against Potassium voltage gated channel KQT-like subfamily, member 2 expressed in HEK 293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RJ4K66PubMed