Found 2 Enz. Inhib. hit(s) with Target = 'Prolyl endopeptidase' and Ligand = 'BDBM50431227' TargetProlyl endopeptidase(Homo sapiens (Human))
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Affinity DataKi: 0.730nMAssay Description:Competitive inhibition of human PREP using Suc-GP-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetProlyl endopeptidase(Homo sapiens (Human))
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human PREP using Z-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
