Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Prolyl endopeptidase FAP' and Ligand = 'BDBM50228403'
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Dainippon Sumitomo Pharma Co., Ltd

Curated by ChEMBL
LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Inhibition of FAPalphaMore data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of recombinant mouse FAP purified from HEK293 cell supernatant using Ala-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp

Curated by ChEMBL
LigandPNGBDBM50228403((R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-met...)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair