Found 4 Enz. Inhib. hit(s) with Target = 'Prolyl endopeptidase FAP' and Ligand = 'BDBM50431242' TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Competitive inhibition of human FAP using Suc-GP-AMC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant mouse FAP purified from HEK293 cell supernatant using Ala-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
TargetProlyl endopeptidase FAP(Homo sapiens (Human))
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Tufts University Sackler School of Biomedical Sciences
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of human FAP using Z-Gly-Pro-AMC as substrate preincubated for 10 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
