Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Prolyl endopeptidase FAP' and Ligand = 'BDBM50434159'
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434159(CHEMBL2385277 | US9346814, Ref Cmpd No 7 (example ...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KP83J7PubMed
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
University of Antwerp (UA)

Curated by ChEMBL
LigandPNGBDBM50434159(CHEMBL2385277 | US9346814, Ref Cmpd No 7 (example ...)copy SMILEScopy InChI
Affinity DataIC50: 420nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W37V6DUS Patent