Found 3 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP1 subtype' and Ligand = 'BDBM50085910'
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by PDSP Ki Database
Merck Frosst Centre for Therapeutic Research
Curated by PDSP Ki Database
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by PDSP Ki Database
Merck Frosst Centre for Therapeutic Research
Curated by PDSP Ki Database
Affinity DataIC50: 496nMAssay Description:Affinity for Prostanoid EP1 receptor expressed in COS-7 cells.More data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP1 subtype(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by PDSP Ki Database
Merck Frosst Centre for Therapeutic Research
Curated by PDSP Ki Database
Affinity DataEC50: 760nMAssay Description:Functional activity in RAT-1cells, transiently-transfected with human Prostaglandin E receptor EP1 (% of control ligand, 17-phi-PGE2=80%)More data for this Ligand-Target Pair