Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-5' and Ligand = 'BDBM50434762'
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina

Curated by ChEMBL
LigandPNGBDBM50434762(CHEMBL2385818)copy SMILEScopy InChI
Affinity DataKi:  1.34E+3nMAssay Description:Inhibition of human 20S proteasome chymotrypsin like activity using Suc-Leu-Leu-Val-Tyr-AMC as substrate measured over 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46TC8PubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ degli Studi di Messina

Curated by ChEMBL
LigandPNGBDBM50434762(CHEMBL2385818)copy SMILEScopy InChI
Affinity DataKi:  1.34E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome beta 5 subunit assessed as Suc-Leu-Leu-Val-Tyr-AMC substrate hydrolysis after 10 min...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N24XMPubMed