Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-5' and Ligand = 'BDBM50450706'
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Heinrich Heine University D£sseldorf

Curated by ChEMBL
LigandPNGBDBM50450706(CHEMBL4167623)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human HL60 cells using Suc-LLVY aminoluciferin as substrate after 2 hrs by proteasome-G...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9DMWPubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Heinrich Heine University D£sseldorf

Curated by ChEMBL
LigandPNGBDBM50450706(CHEMBL4167623)copy SMILEScopy InChI
Affinity DataIC50: 394nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in human SEM cells using Suc-LLVY aminoluciferin as substrate after 2 hrs by proteasome-Gl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9DMWPubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Heinrich Heine University D£sseldorf

Curated by ChEMBL
LigandPNGBDBM50450706(CHEMBL4167623)copy SMILEScopy InChI
Affinity DataIC50: 821nMAssay Description:Inhibition of chymotrypsin-like activity of 20S proteasome in imatinib-resistant human SUP-B15 cells using Suc-LLVY aminoluciferin as substrate after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9DMWPubMed