Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Protein cereblon' and Ligand = 'BDBM50088517'
TargetProtein cereblon(Homo sapiens (Human))TBA
LigandPNGBDBM50088517(CHEBI:16704 | Uridine)copy SMILEScopy InChI
Affinity DataKi:  3.90E+5nMAssay Description:Binding affinity to human CRBN-thalidomide binding domain expressed in Escherichia coli by measuring baseline corrected normalized fluorescence by MS...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J1BPubMed
TargetProtein cereblon(Homo sapiens (Human))TBA
LigandPNGBDBM50088517(CHEBI:16704 | Uridine)copy SMILEScopy InChI
Affinity DataIC50: 7.57E+5nMAssay Description:Binding affinity to human CRBN-thalidomide binding domain expressed in Escherichia coli by measuring baseline corrected normalized fluorescence by MS...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J1BPubMed