Found 15 Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha type' and Ligand = 'BDBM3149' TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 0.0740nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Protein kinase C etaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibitory concentration against recombinant human Protein kinase C alpha isozymeMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of Protein kinase C beta 2More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of protein kinase C beta IMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of protein kinase C gammaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 74nMpH: 7.5 T: 2°CAssay Description:The activity of PKC, activated by phosphatidylerine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich his...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 74nMpH: 7.5 T: 2°CAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of California at San Diego
Curated by ChEMBL
University of California at San Diego
Curated by ChEMBL
Affinity DataKd: 6.40nMAssay Description:Binding affinity to PKCalpha (unknown origin) using Lys-Arg-Thr-Leu-Arg-Arg as substrate after 8 mins in presence of [gamma-32P]ATP by liquid scintil...More data for this Ligand-Target Pair
