Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha type' and Ligand = 'BDBM50059769'
TargetProtein kinase C alpha type(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50059769(CHEMBL3393745)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [20-3H] phorbol 12, 13-dibutylate from recombinant PKCalpha (unknown origin) in presence of 100 ug/ml 100% phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930VV0PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50059769(CHEMBL3393745)copy SMILEScopy InChI
Affinity DataKi:  116nMAssay Description:Displacement of [20-3H] phorbol 12, 13-dibutylate from recombinant PKCalpha (unknown origin) in presence of nuclear membrane mimetic lipid mixtureMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930VV0PubMed