Found 2 Enz. Inhib. hit(s) with Target = 'Protein kinase C theta type' and Ligand = 'BDBM50427363' TargetProtein kinase C theta type(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Inhibition of full-length recombinant PKC theta (unknown origin) using ERMRPRKRQGSVRRRV as substrate after 60 mins by scintillation counting analysis...More data for this Ligand-Target Pair
TargetProtein kinase C theta type(Homo sapiens (Human))
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Vertex Pharmaceuticals (Europe) Ltd.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of full-length recombinant PKC theta (unknown origin) using ERMRPRKRQGSVRRRV as substrate after 60 mins by scintillation counting analysis...More data for this Ligand-Target Pair
