Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Protein kinase C zeta type' and Ligand = 'BDBM50542096'
TargetProtein kinase C zeta type(Homo sapiens (Human))TBA
LigandPNGBDBM50542096(CHEMBL4637961)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22XQPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))TBA
LigandPNGBDBM50542096(CHEMBL4637961)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed